Development of the First Two-Pore Domain Potassium Channel TWIK-Related K+ Channel 1-Selective Agonist Possessing in Vivo Antinociceptive Activity.

J Med Chem. 2017 Feb 9;60(3):1076-1088. doi: 10.1021/acs.jmedchem.6b01285. Epub 2017 Jan 20. Vivier D1, Soussia IB2, Rodrigues N1, Lolignier S3, Devilliers M3, Chatelain FC2, Prival L3, Chapuy E3, Bourdier G1, Bennis K1, Lesage F2, Eschalier A3,4, Busserolles J3, Ducki S1.